Rapid synthesis a thousand times

Rapid synthesis a thousand times

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Access through your institution Buy or subscribe A robotic system that can carry out and analyse 1,536 chemical reactions in less than a day could help to accelerate drug discovery. Tim Cernak and Spencer Dreher at pharmaceutical company Merck in Massachusetts and New Jersey and their colleagues used the system to couple a model substrate with 16 other molecules, in combination with 16 different palladium catalysts and 6 basic reagents. Each of these unique mixtures was dissolved in 1 microlitre of solvent, automatically dispensed into a separate chamber on a 1,536-well plate, and its products were analysed to determine optimum reaction conditions. This is a preview of subscription content, access via your institution ACCESS OPTIONS Access through your institution Subscribe to this journal Receive 51 print issues and online access $199.00 per year only $3.90 per issue Learn more Buy this article * Purchase on SpringerLink * Instant access to full article PDF Buy now Prices may be subject to local taxes which are calculated during checkout ADDITIONAL ACCESS OPTIONS: * Log in * Learn about institutional subscriptions * Read our FAQs * Contact customer support RIGHTS AND PERMISSIONS Reprints and permissions ABOUT THIS ARTICLE CITE THIS ARTICLE Rapid synthesis a thousand times. _Nature_ 515, 468 (2014). https://doi.org/10.1038/515468d Download citation * Published: 26 November 2014 * Issue Date: 27 November 2014 * DOI: https://doi.org/10.1038/515468d SHARE THIS ARTICLE Anyone you share the following link with will be able to read this content: Get shareable link Sorry, a shareable link is not currently available for this article. Copy to clipboard Provided by the Springer Nature SharedIt content-sharing initiative

Access through your institution Buy or subscribe A robotic system that can carry out and analyse 1,536 chemical reactions in less than a day could help to accelerate drug discovery. Tim


Cernak and Spencer Dreher at pharmaceutical company Merck in Massachusetts and New Jersey and their colleagues used the system to couple a model substrate with 16 other molecules, in


combination with 16 different palladium catalysts and 6 basic reagents. Each of these unique mixtures was dissolved in 1 microlitre of solvent, automatically dispensed into a separate


chamber on a 1,536-well plate, and its products were analysed to determine optimum reaction conditions. This is a preview of subscription content, access via your institution ACCESS OPTIONS


Access through your institution Subscribe to this journal Receive 51 print issues and online access $199.00 per year only $3.90 per issue Learn more Buy this article * Purchase on


SpringerLink * Instant access to full article PDF Buy now Prices may be subject to local taxes which are calculated during checkout ADDITIONAL ACCESS OPTIONS: * Log in * Learn about


institutional subscriptions * Read our FAQs * Contact customer support RIGHTS AND PERMISSIONS Reprints and permissions ABOUT THIS ARTICLE CITE THIS ARTICLE Rapid synthesis a thousand times.


_Nature_ 515, 468 (2014). https://doi.org/10.1038/515468d Download citation * Published: 26 November 2014 * Issue Date: 27 November 2014 * DOI: https://doi.org/10.1038/515468d SHARE THIS


ARTICLE Anyone you share the following link with will be able to read this content: Get shareable link Sorry, a shareable link is not currently available for this article. Copy to clipboard


Provided by the Springer Nature SharedIt content-sharing initiative